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Table 4D CNS Diseases/Clinical Situations in Which First-Generation H1 Antihistamines Are Used*

From: H1 Antihistamines: Current Status and Future Directions

Insomnia

Perioperative sedation

Antiemetic effect

Analgesia

Akathisia

Serotonin syndrome

Anxiety

Migraine headache

  1. *Safer alternatives are preferred.